Electrophile-driven regioselective synthesis of functionalized quinolines | |
Department | 固体润滑国家重点实验室 |
Ali Shaukat; Zhu HT(祝海涛); Xia XF(夏晓峰); Ji KG(纪克攻); Yang YF(杨艳芳); Song XR(宋贤荣); Liang YM(梁永民); Liang YM(梁永民) | |
2011 | |
Source Publication | J. Org. Lett. |
ISSN | 0022-3263 |
Volume | 13Issue:10Pages:2598-2601 |
Abstract | Highly substituted 3-iodoquinolines bearing different alkyl and aryl moieties can be synthesized in moderate to excellent yields (up to 99%) by 6-endo-dig iodocyclization of 2-tosylaminophenylprop-1-yn-3-ols with molecular iodine (I2) under mild conditions. The cyclization is highly regioselective and the resulting 3-iodoquinolines can be further functionalized by various coupling reactions. |
Subject Area | 材料科学与物理化学 |
Funding Organization | the National Science Foundation (NSF-21072080);the National Basic Research Program of China (973 Program),2010CB833203 |
Indexed By | SCI |
Language | 英语 |
Citation statistics | |
Document Type | 期刊论文 |
Identifier | http://ir.licp.cn/handle/362003/3963 |
Collection | 固体润滑国家重点实验室(LSL) |
Corresponding Author | Liang YM(梁永民) |
Recommended Citation GB/T 7714 | Ali Shaukat,Zhu HT,Xia XF,et al. Electrophile-driven regioselective synthesis of functionalized quinolines[J]. J. Org. Lett.,2011,13(10):2598-2601. |
APA | Ali Shaukat.,Zhu HT.,Xia XF.,Ji KG.,Yang YF.,...&梁永民.(2011).Electrophile-driven regioselective synthesis of functionalized quinolines.J. Org. Lett.,13(10),2598-2601. |
MLA | Ali Shaukat,et al."Electrophile-driven regioselective synthesis of functionalized quinolines".J. Org. Lett. 13.10(2011):2598-2601. |
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20112598-2601.PDF(752KB) | 期刊论文 | 出版稿 | 开放获取 | CC BY-NC-SA | View Application Full Text |
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